Collect. Czech. Chem. Commun.
1991, 56, 2978-2985
https://doi.org/10.1135/cccc19912978
Correlation of structural parameters with antituberculotic activity in a group of 2-benzamidobenzothiazoles
Karel Waissera, Jiří Kuneša and Želmíra Odlerováb
a Department of Inorganic and Organic Chemistry, Pharmaceutical Faculty, Charles University, 501 65 Hradec Králové
b Research Institute of Preventive and Clinical Medicine, 833 01 Bratislava
Individual author index pages
Other CCCC articles of these authors
- Vojtěch Balšánek, Lucie Tichotová, Jiří Kuneš, Marcel Špulák, Milan Pour*, Ivan Votruba and Vladimír Buchta
Cytostatic tetrazole–butenolide conjugates: linking tetrazole and butenolide rings via stille coupling and biological activity of the target substances
2009, Vol. 74, Issue 7-8, pp. 1161–1178 [Abstract] - Marta Kučerová-Chlupáčová, Veronika Opletalová*, Josef Jampílek, Jan Doležel, Jiří Dohnal, Milan Pour, Jiří Kuneš and Viktor Voříšek
New Hydrophobicity Constants of Substituents in Pyrazine Rings Derived from RP-HPLC Study
2008, Vol. 73, Issue 1, pp. 1–18 [Abstract] - Ivan Šnajdr, Jan Pavlík, Radan Schiller, Jiří Kuneš and Milan Pour*
Pentenolide Analogues of Antifungal Butenolides: Strategies Towards 3,6-Disubstituted Pyranones and Unexpected Loss of Biological Effect
2007, Vol. 72, Issue 11, pp. 1472–1498 [Abstract] - Veronika Opletalová*, Milan Pour, Jiří Kuneš, Vladimír Buchta, Luís Silva, Katarína Kráľová, Marta Chlupáčová, Dana Meltrová, Milan Peterka and Martina Posledníková
Synthesis and Biological Evaluation of (E)-3-(Nitrophenyl)-1-(pyrazin-2-yl)prop-2-en-1-ones
2006, Vol. 71, Issue 1, pp. 44–58 [Abstract] - Karel Waisser*, Milan Peřina, Věra Klimešová and Jarmila Kaustová
On the Relationship between the Structure and Antimycobacterial Activity of Substituted N-Benzylsalicylamides
2003, Vol. 68, Issue 7, pp. 1275–1294 [Abstract] - Jiří Kuneš, Vojtěch Balšánek, Milan Pour* and Vladimír Buchta
Synthesis and Antifungal Activity Evaluation of 3-Hetaryl-2,5-dihydrofuran-2-ones. An Unusual Fragmentation of the Oxazole Ring via 2,3-Selenoxide Shift
2001, Vol. 66, Issue 12, pp. 1809–1830 [Abstract] - Karel Waisser*, Miloš Macháček, Hynek Dostál, Jiří Gregor, Lenka Kubicová, Věra Klimešová, Jiří Kuneš, Karel Palát, Jr., Jana Hladůvková, Jarmila Kaustová and Ute Möllmann
Relationships Between the Chemical Structure of Substances and Their Antimycobacterial Activity Against Atypical Strains. Part 18. 3-Phenyl-2H-1,3-benzoxazine-2,4(3H)-diones and Isosteric 3-Phenylquinazoline-2,4(1H,3H)-diones
1999, Vol. 64, Issue 11, pp. 1902–1924 [Abstract] - Miroslav Holík*, Zdeněk Friedl, Karel Waisser and Jiří Gregor
Multivariate Regression with Substituent Shift Increments. IV. 2-(4-X-Phenyl)-1,3-dihydro-2H-isoindole-1,3-diones and 3-(4-X-Phenyl)-3,4-dihydro-2H-1,3-benzoxazine-2,4-diones
1999, Vol. 64, Issue 10, pp. 1709–1726 [Abstract] - Karel Waisser*, Karel Palát, Jr. and Otto Exner*
Substituent Effects on Conformational Equilibria: Substituted Thiobenzanilides
1999, Vol. 64, Issue 8, pp. 1295–1306 [Abstract] - Věra Klimešová*, Martin Svoboda, Karel Waisser, Milan Pour and Jarmila Kaustová
Synthesis and Antimicrobial Activity of New 4-(Benzylsulfanyl)pyridine Derivatives
1999, Vol. 64, Issue 2, pp. 417–434 [Abstract] - Václav Kozmík, Pavel Lhoták, Želmíra Odlerová and Jaroslav Paleček
Azachalcone Derivatives and Their Bis Substituted Analogs as Novel Antimycobacterial Agents
1998, Vol. 63, Issue 5, pp. 698–712 [Abstract] - Jiří Kuneš, Jiří Jáchym, Petr Jirásko, Želmíra Odlerová and Karel Waisser
Combination of the Topliss Approach with the Free-Wilson Analysis in the Study of Antimycobacterial Activityof 4-Alkylthiobenzanilides
1997, Vol. 62, Issue 9, pp. 1503–1510 [Abstract] - Katarína Kráľová, František Šeršeň, Věra Klimešová and Karel Waisser
Effect of 2-Alkylthio-4-pyridinecarbothiamides on Photosynthetic Electron Transport in Spinach Chloroplasts
1997, Vol. 62, Issue 3, pp. 516–520 [Abstract] - Hans-Dietrich Stachel, Želmíra Odlerová and Karel Waisser
A New Pharmacophore of Potential Antimycobacterial Activity: The Disulfide Group in the Ring of Alicyclic Compounds
1997, Vol. 62, Issue 3, pp. 510–515 [Abstract] - Jiří Hartl, Martin Doležal, Jana Krinková, Antonín Lyčka and Želmíra Odlerová
Synthesis and Antituberculotic Activity of 5-Alkyl-6-chloro-2-pyrazinecarboxamides and Corresponding Thioamides
1996, Vol. 61, Issue 7, pp. 1109–1114 [Abstract] - Martin Doležal, Jiří Hartl, Antonín Lyčka, Vladimír Buchta and Želmíra Odlerová
Synthesis and Antituberculotic Properties of Some Substituted Pyrazinecarbothioamides
1996, Vol. 61, Issue 7, pp. 1102–1108 [Abstract] - Karel Waisser, Jiří Kuneš, Alexandr Hrabálek, Miloš Macháček and Želmíra Odlerová
New Groups of Potential Antituberculotics: 5-Alkylthio-1-aryltetrazoles
1996, Vol. 61, Issue 5, pp. 791–798 [Abstract] - Martin Doležal, Jiří Hartl, Antonín Lyčka, Vladimír Buchta and Želmíra Odlerová
Synthesis and Antituberculotic Activity of Some Substituted 3-Arylamino-5-cyano-2-pyrazinecarboxamides
1995, Vol. 60, Issue 7, pp. 1236–1241 [Abstract] - Karel Waisser, Jiří Kuneš, Alexandr Hrabálek and Želmíra Odlerová
New Groups of Potential Antituberculotics: Bis(1-aryltetrazol-5-yl) Disulfides. Structure Activity Relationship
1994, Vol. 59, Issue 1, pp. 234–238 [Abstract] - Karel Waisser, Lenka Kubicová, Věra Klimešová and Želmíra Odlerová
New Groups of Potential Antituberculotics: 3-Aryl-2H,4H-benz[e][1,3]oxazine-2,4-diones. Comparison of the Topliss Approach with Regression Analysis
1993, Vol. 58, Issue 12, pp. 2977–2982 [Abstract] - Karel Waisser, Lenka Kubicová and Želmíra Odlerová
Antituberculotic 4'-Cyclohexylthiobenzanilides: Combination of Free-Wilson Method in QSAR with Topliss Approach
1993, Vol. 58, Issue 1, pp. 205–212 [Abstract] - Karel Waisser, Miloš Macháček, Želmíra Odlerová, Wilfried Thiel and Roland Mayer
Antimycobacterial 2-Arylamino-2-Thioxoacetamides
1993, Vol. 58, Issue 1, pp. 197–204 [Abstract] - Karel Waisser, Jiří Kuneš, Jiří Klimeš, Miroslav Polášek and Želmíra Odlerová
Relations between Structure and Antituberculotic Activity of 4-Alkoxybenzoic Acids
1993, Vol. 58, Issue 1, pp. 191–196 [Abstract] - Miroslav Polášek, Karel Waisser and Tomáš Bouček
Determination of the substituent constant σp- for the thioamide group -CSNH2 from the ionization of anilines and phenols
1991, Vol. 56, Issue 12, pp. 2964–2968 [Abstract] - Karel Waisser and Jana Bořková
Relations between structure and antituberculotic activity in a group of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1991, Vol. 56, Issue 11, pp. 2395–2401 [Abstract] - Karel Waisser, Jiří Vanžura, Alexandr Hrabálek, Jarmila Vinšová, Štefan Grešák, Jiří Hruška and Želimíra Odlerová
Antimycobacterial derivatives of tetrazole
1991, Vol. 56, Issue 11, pp. 2389–2394 [Abstract] - Karel Dlabal, Karel Palát, Antonín Lyčka and Želmíra Odlerová
Synthesis and 1H and 13C NMR spectra of sulfur derivatives of pyrazine derived from amidation product of 2-chloropyrazine and 6-chloro-2-pyrazinecarbonitrile. Tuberculostatic activity
1990, Vol. 55, Issue 10, pp. 2493–2501 [Abstract] - Karel Waisser, Nestor Houngbedji, Miloš Macháček, Miroslav Sekera, Josef Urban and Želmíra Odlerová
Antimycobacterial thiobenzanilides
1990, Vol. 55, Issue 1, pp. 307–316 [Abstract] - Naďa Zimová, Ivan Němec, Miroslava Ehlová and Karel Waisser
The effect of the structure of the substituent in position ten on the voltammetric behaviour of phenothiazin derivatives
1990, Vol. 55, Issue 1, pp. 63–71 [Abstract] - Karel Waisser, Miloš Macháček, Jean Lebvoua, Jiří Hrbata and Jaroslav Dršata
Quantitative relations between chemical structure and hepatotoxicity of thiobenzamides
1988, Vol. 53, Issue 11, pp. 2957–2961 [Abstract] - Otto Exner and Karel Waisser
Dipole moment and electron distribution of the thioamide group
1982, Vol. 47, Issue 3, pp. 828–837 [Abstract]